SCHEMBL7514845

SCHEMBL7514845

Nc1ncc(Sc2c(Cl)cccc2Cl)c(=O)[nH]1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TYMS P04818 8/20 0.42
DHFR P00374 1/20 0.42
PTPN11 Q06124 4/20 0.39
XDH P47989 2/20 0.36
MAPK14 Q16539 1/20 0.35
AOC3 Q16853 1/20 0.35
MASP2 O00187 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7512558 0.78 RXFP1 (0.50) TYMSDHFRXDH
SCHEMBL7515297 0.78 ITGB2 (0.50) TYMSDHFRPTPN11XDHMAPK14
SCHEMBL7519197 0.76 MAPK11 (0.41) TYMSPTPN11MAPK14
SCHEMBL7515639 0.76 TYMS (0.51) TYMSDHFRXDHAOC3MASP2
SCHEMBL7518203 0.73 TYMS (0.37) TYMSXDHMAPK14
SCHEMBL6049582 0.72 NUDT1 (0.50) TYMSPTPN11XDH
SCHEMBL7515343 0.72 TYMS (0.42) TYMSDHFRXDH
SCHEMBL11543373 0.72
SCHEMBL23339220 0.71 NOS1 (0.40) TYMSXDHAOC3MASP2
SCHEMBL7518650 0.69 TYMS (0.43) TYMSDHFRAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165522-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP disclosed
WO-2000059893-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-12 WO disclosed