SCHEMBL7512558

SCHEMBL7512558

Nc1ncc(Sc2ccc(Cl)cc2)c(=O)[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.50
TYMS P04818 5/20 0.48
DHFR P00374 3/20 0.46
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
EGFR P00533 1/20 0.41
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.40
PKM P14618 1/20 0.40
RHEB Q15382 2/20 0.40
LTA4H P09960 1/20 0.40
HAO1 Q9UJM8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
XDH P47989 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515639 0.85 TYMS (0.51) TYMSDHFRXDH
SCHEMBL7515343 0.84 TYMS (0.42) RXFP1TYMSDHFREGFRLMNA
SCHEMBL7515297 0.81 ITGB2 (0.50) TYMSDHFRALDH1A1CYP1A2CYP3A4
SCHEMBL7524669 0.81 TYMS (0.51) TYMSDHFRALDH1A1HAO1XDH
SCHEMBL7518650 0.81 TYMS (0.43) TYMSDHFR
SCHEMBL7518203 0.79 TYMS (0.37) TYMSHPGDLMNALTA4HXDH
SCHEMBL7514845 0.78 TYMS (0.42) TYMSDHFRXDH
SCHEMBL7519197 0.73 MAPK11 (0.41) TYMSKDM4EL3MBTL1
SCHEMBL7708406 0.72 LTA4H (0.50) RXFP1KDM4EALDH1A1CYP1A2HPGD
SCHEMBL23339220 0.71 NOS1 (0.40) TYMSKDM4EALDH1A1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165522-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP disclosed
WO-2000059893-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-12 WO disclosed