SCHEMBL7518650

SCHEMBL7518650

CCc1ccc(Sc2cnc(N)[nH]c2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TYMS P04818 16/20 0.43
DHFR P00374 7/20 0.41
AOC3 Q16853 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515343 0.84 TYMS (0.42) TYMSDHFR
SCHEMBL7515639 0.82 TYMS (0.51) TYMSDHFRAOC3
SCHEMBL7512558 0.81 RXFP1 (0.50) TYMSDHFR
SCHEMBL7524669 0.77 TYMS (0.51) TYMSDHFR
SCHEMBL5204052 0.71 SMN1; SMN2 (0.42) TYMS
SCHEMBL23339220 0.71 NOS1 (0.40) TYMSAOC3
SCHEMBL13039021 0.69 NOS1 (0.42) TYMSDHFRAOC3
SCHEMBL7514845 0.69 TYMS (0.42) TYMSDHFRAOC3
SCHEMBL3445980 0.66
SCHEMBL7515297 0.66 ITGB2 (0.50) TYMSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165522-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP disclosed
WO-2000059893-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-12 WO disclosed