SCHEMBL751493

SCHEMBL751493

Cc1ccc(S(=O)(=O)C(Br)(Br)Br)c([N+](=O)[O-])c1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
CYP3A4 P08684 1/20 0.55
MCOLN3 Q8TDD5 1/20 0.51
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NFKBIA P25963 2/20 0.44
RELA Q04206 2/20 0.44
AGTR1 P30556 1/20 0.44
OPRK1 P41145 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
GPR35 Q9HC97 1/20 0.42
THRB P10828 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KAT2B Q92831 2/20 0.39
VCAM1 P19320 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL751494 1.00 TSHR (0.55) TSHRCYP3A4MCOLN3MEN1KMT2A
SCHEMBL15356391 0.88 TSHR (0.56) TSHRCYP3A4MCOLN3MEN1KMT2A
SCHEMBL21137711 0.83 TSHR (0.50) TSHRCYP3A4MCOLN3MEN1KMT2A
SCHEMBL4067424 0.81 TSHR (0.60) TSHRCYP3A4MCOLN3MEN1KMT2A
SCHEMBL10619019 0.81 TSHR (0.60) TSHRCYP3A4MCOLN3MEN1KMT2A
SCHEMBL752795 0.80 KIF18A (0.59) TSHRALDH1A1VCAM1
SCHEMBL752794 0.80 KIF18A (0.59) TSHRALDH1A1VCAM1
SCHEMBL137704 0.79 TSHR (0.58) TSHRCYP3A4MCOLN3MEN1KMT2A
SCHEMBL11119285 0.79 TSHR (0.58) TSHRCYP3A4MCOLN3MEN1KMT2A
SCHEMBL4807396 0.79 TSHR (0.58) TSHRCYP3A4MCOLN3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2213166-B1 Biocidal compounds containing 2-methylisothiazolin-3-one and a haloalkylsulfone THOR GMBH (DE) 2012-03-21 EP claimed
EP-2213166-A1 Biocidal compounds containing 2-methylisothiazolin-3-one and a haloalkylsulfone THOR GmbH (DE) 2010-08-04 EP claimed
US-20100189811-A1 Biocide compositions comprising 3-methylisothiazolin-3-one and a haloalkyl sulphone THOR GMBH (DE) 2010-07-29 US claimed
EP-2216372-B1 Compounds for preventing Ghost odour THOR GMBH (DE) 2014-06-04 EP disclosed
US-8287631-B2 Compounds for preventing ghost odour THOR GMBH (DE) 2012-10-16 US disclosed
EP-2213166-B1 Biocidal compounds containing 2-methylisothiazolin-3-one and a haloalkylsulfone THOR GMBH (DE) 2012-03-21 EP disclosed
EP-2216372-A1 Compounds for preventing Ghost odour THOR GmbH (DE) 2010-08-11 EP disclosed
EP-2213166-A1 Biocidal compounds containing 2-methylisothiazolin-3-one and a haloalkylsulfone THOR GmbH (DE) 2010-08-04 EP disclosed
US-20100186631-A1 Compounds for preventing ghost odour THOR GMBH (DE) 2010-07-29 US disclosed
US-20100189811-A1 Biocide compositions comprising 3-methylisothiazolin-3-one and a haloalkyl sulphone THOR GMBH (DE) 2010-07-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100189811-A1 Biocide compositions comprising 3-methylisothiazolin-3-one and a haloalkyl sulphone MBTD1, MPST, B2M TSHR 4791/4885CYP3A4 1279/4885MCOLN3 447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.