SCHEMBL751497

SCHEMBL751497

O=C(COC(=O)C1CCCN1C(=O)O)c1ccc2c(c1)COCc1cc(Br)ccc1-2

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
SRD5A1 P18405 1/20 0.37
SRD5A2 P31213 1/20 0.37
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
FKBP1A P62942 8/20 0.36
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL750978 0.91 SRD5A1 (0.47) ALDH1A1SRD5A1SRD5A2MAPTTDP1
SCHEMBL2706884 0.88 USP30 (0.42) ALDH1A1KMT2A
SCHEMBL204193 0.88 USP30 (0.42) ALDH1A1KMT2A
SCHEMBL749960 0.83 ALDH1A1 (0.44) ALDH1A1MAPTTDP1FKBP1AKMT2A
SCHEMBL2757491 0.83 ALDH1A1 (0.44) ALDH1A1MAPTTDP1FKBP1AKMT2A
SCHEMBL18462759 0.81 NPC1 (0.46) ALDH1A1KMT2AL3MBTL1
SCHEMBL2706099 0.81 NPC1 (0.46) ALDH1A1KMT2AL3MBTL1
SCHEMBL751808 0.81 ALDH1A1 (0.41) ALDH1A1MAPTTDP1FKBP1AKMT2A
SCHEMBL203386 0.79 NPC1 (0.42) ALDH1A1KMT2A
SCHEMBL2708423 0.79 NPC1 (0.42) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed