SCHEMBL7517281

SCHEMBL7517281

NS(=O)(=O)c1ccc(NC(=O)NC2=CC(=O)SC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.62
CA12 O43570 16/20 0.56
CA1 P00915 16/20 0.56
CA2 P00918 16/20 0.56
CA9 Q16790 16/20 0.56
MEN1 O00255 2/20 0.55
CA4 P22748 1/20 0.55
CA7 P43166 1/20 0.55
PTPN7 P35236 1/20 0.55
MAPT P10636 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7563850 0.81 PIP4K2A (0.45) KMT2AMEN1
SCHEMBL8210609 0.80 RAB9A (0.50) KMT2AMEN1PTPN7MAPT
SCHEMBL7518699 0.80 MAOA (0.51) KMT2ACA12CA1CA2CA9
SCHEMBL7529461 0.80 KMT2A (0.49) KMT2ACA12CA1CA2CA9
SCHEMBL7521962 0.80 ALDH1A1 (0.51) KMT2ACA12CA1CA2CA9
SCHEMBL7524755 0.80 SMN1; SMN2 (0.55) KMT2AMEN1MAPT
SCHEMBL28499329 0.79 KMT2A (1.00) KMT2ACA12CA1CA2CA9
SCHEMBL7522234 0.76 KMT2A (0.62) KMT2ACA12CA1CA2CA9
SCHEMBL7518438 0.74 EPHX1 (0.61) KMT2ACA2CA9MEN1CA4
SCHEMBL6252334 0.73 KMT2A (1.00) KMT2ACA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020058694-A1 Ureido and thioureido derivatives of 4-amino-2(5H)-furanones and 4-amino-2(5H)-thiophenones as antitumor agents ROCHE DIAGNOSTICS GMBH 2002-05-16 US disclosed
US-6333346-B1 AMINOFURANONEUREAS OR THIOUREAS 4-AMINO-2(5H)-THIOPHENONES AS ANTITUMOR AGENTS ROCHE DIAGNOSTICS GMBH (DE) 2001-12-25 US disclosed
EP-1009747-A1 UREIDO AND THIOUREIDO DERIVATIVES OF 4-AMINO-2(5H)-FURANONES AND 4-AMINO-2(5H)-THIOPHENONES AS ANTITUMOR AGENTS Roche Diagnostics GmbH (DE) 2000-06-21 EP disclosed
WO-1999012917-A1 UREIDO AND THIOUREIDO DERIVATIVES OF 4-AMINO-2(5H)-FURANONES AND 4-AMINO-2(5H)-THIOPHENONES AS ANTITUMOR AGENTS ROCHE DIAGNOSTICS GMBH (DE) 1999-03-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020058694-A1 Ureido and thioureido derivatives of 4-amino-2(5H)-furanones and 4-amino-2(5H)-thiophenones as antitumor agents UTS2R, SRD5A2, SRD5A1 KMT2A 3288/4885CA12 3070/4885CA1 2207/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.