SCHEMBL7517995

SCHEMBL7517995

CCCCCCCCc1ccc2c(c1)nc(F)c1cc(O)ccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.49
PTGS2 P35354 4/20 0.49
ESR1 P03372 2/20 0.49
ADRA2A P08913 2/20 0.49
ADORA3 P0DMS8 2/20 0.49
TACR2 P21452 2/20 0.49
SLC6A2 P23975 2/20 0.49
SLC6A4 P31645 2/20 0.49
SLC6A3 Q01959 2/20 0.49
TP53 P04637 2/20 0.49
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
HSD17B10 Q99714 2/20 0.49
LMNA P02545 1/20 0.49
SHBG P04278 1/20 0.49
HSPD1 P10809 1/20 0.49
ADRB3 P13945 1/20 0.49
HTR2C P28335 1/20 0.49
HSPE1 P61604 1/20 0.49
HIF1A Q16665 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7524265 0.95 CYP3A4 (0.49) CYP3A4PTGS2ESR1ADRA2AADORA3
SCHEMBL7523369 0.82 EIF4A1 (0.41) CYP3A4PTGS2ESR1ADRA2AADORA3
SCHEMBL7528065 0.81 MAPK1 (0.41) CYP3A4TP53KDM4EALDH1A1LMNA
SCHEMBL19625906 0.79 TLR8 (0.50) CYP3A4PTGS2ESR1ADRA2AADORA3
SCHEMBL7519044 0.78 NR5A1 (0.51) ALDH1A1MAPTMEN1KMT2AGAA
SCHEMBL7561109 0.76 PTGS2 (0.51) CYP3A4PTGS2ESR1ADRA2AADORA3
SCHEMBL7515612 0.76 CYP3A4 (0.41) CYP3A4ALDH1A1HSD17B10LMNAMAPT
SCHEMBL7519026 0.76 S1PR1 (0.37) CYP3A4ALDH1A1LMNAMEN1KMT2A
SCHEMBL2050474 0.73 PTGS2 (0.67) CYP3A4PTGS2ESR1ADRA2AADORA3
SCHEMBL9700041 0.73 PTGS2 (0.67) CYP3A4PTGS2ESR1ADRA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946513-B1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES AVENTIS RES & TECH GMBH & CO (DE) 2002-01-30 EP disclosed
US-6120703-A Derivatives of 6-fluorophenanthridine for liquid crystal mixtures AVENTIS RESEARCH & TECHNOLOGIES DEUTSCHLAND GMBH & CO. KG (DE) 2000-09-19 US disclosed
EP-0946513-A1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES Aventis Research & Technologies GmbH & Co. KG (DE) 1999-10-06 EP disclosed
WO-1998027060-A1 DERIVATIVES OF 6-FLUOROPHENANTHRIDINE FOR LIQUID CRYSTAL MIXTURES AVENTIS RESEARCH & TECHNOLOGIES GMBH & CO KG (DE) 1998-06-25 WO disclosed