SCHEMBL7518286

SCHEMBL7518286

CC(=O)N1CCN(c2nc(N)ncc2Sc2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EIF2AK4 Q9P2K8 1/20 0.46
DHFR P00374 2/20 0.42
MET P08581 1/20 0.42
AKT1 P31749 1/20 0.41
AKT2 P31751 1/20 0.41
AKT3 Q9Y243 1/20 0.41
TRPV1 Q8NER1 3/20 0.41
ABL1 P00519 1/20 0.41
BCR P11274 1/20 0.41
P2RX3 P56373 1/20 0.41
CNR2 P34972 1/20 0.40
ITGB2 P05107 1/20 0.40
ICAM1 P05362 1/20 0.40
ITGAL P20701 1/20 0.40
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
TRPA1 O75762 1/20 0.39
SCN9A Q15858 1/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7508846 0.87 RXFP1 (0.44) DHFRAKT1AKT2AKT3LMNA
SCHEMBL7519963 0.87 CKS1B (0.46) CNR2LMNASMN1; SMN2RXFP1ALDH1A1
SCHEMBL7516894 0.86 RXFP1 (0.55) DHFRAKT1CNR2ITGALLMNA
SCHEMBL7516678 0.86 RXFP1 (0.41) DHFRAKT1AKT2AKT3RXFP1
SCHEMBL7519270 0.85 ALDH1A1 (0.42) LMNASMN1; SMN2HTTRXFP1KMT2A
SCHEMBL7522989 0.78 CNR2 (0.44) DHFRCNR2KMT2A
SCHEMBL7514338 0.77 RXFP1 (0.45) AKT1ITGB2ICAM1ITGALLMNA
SCHEMBL7519326 0.76 ALDH1A1 (0.43) DHFRTRPV1ABL1BCRCNR2
SCHEMBL7512812 0.76 PTPN11 (0.43) AKT1TRPV1ABL1BCRCNR2
SCHEMBL7514586 0.75 ITGAL (0.52) DHFRABL1BCRCNR2ITGB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165522-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP claimed
WO-2000059893-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-12 WO claimed