SCHEMBL7524669

SCHEMBL7524669

Nc1ncc(Sc2ccc(C(F)(F)F)cc2)c(=O)[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 2/20 0.51
DHFR P00374 1/20 0.44
HAO1 Q9UJM8 1/20 0.42
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
COMT P21964 1/20 0.40
ICAM1 P05362 1/20 0.39
SELE P16581 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 1/20 0.39
HTR1A P08908 1/20 0.39
HTR3A P46098 1/20 0.39
DAO P14920 1/20 0.38
NOTUM Q6P988 1/20 0.38
RECQL P46063 1/20 0.37
XDH P47989 1/20 0.37
PARP1 P09874 1/20 0.36
BRAF P15056 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515639 0.82 TYMS (0.51) TYMSDHFRXDH
SCHEMBL7515343 0.81 TYMS (0.42) TYMSDHFRHAO1MEN1KMT2A
SCHEMBL7512558 0.81 RXFP1 (0.50) TYMSDHFRHAO1ALDH1A1MEN1
SCHEMBL7518650 0.77 TYMS (0.43) TYMSDHFR
SCHEMBL5206874 0.71 L3MBTL1 (0.41) TYMSCOMTICAM1SELE
SCHEMBL7514845 0.69 TYMS (0.42) TYMSDHFRXDH
SCHEMBL23339220 0.68 NOS1 (0.40) TYMSALDH1A1MEN1KMT2AXDH
SCHEMBL1374427 0.68 KDM4E (0.37) ALDH1A1MEN1KMT2AXDHPARP1
SCHEMBL10395372 0.68 GRM5 (0.51) DHFRHAO1ALDH1A1MEN1KMT2A
SCHEMBL8982402 0.67 HAO1 (0.50) TYMSDHFRHAO1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165522-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP disclosed
WO-2000059893-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-12 WO disclosed