SCHEMBL7519289

SCHEMBL7519289

C[Si](C)(CCl)c1ccccc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.39
HSD11B1 P28845 2/20 0.37
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
ATM Q13315 1/20 0.37
NOTUM Q6P988 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
HIF1A Q16665 1/20 0.34
HSD17B10 Q99714 1/20 0.34
POLQ O75417 1/20 0.34
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 2/20 0.34
HTT P42858 1/20 0.34
POLB P06746 2/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30626928 0.81 HSD11B1 (0.42) IDO1HSD11B1ALDH1A1NOTUMCYP1A2
SCHEMBL2295972 0.81 HSD11B1 (0.42) IDO1HSD11B1ALDH1A1NOTUMCYP1A2
SCHEMBL9563607 0.78 HSD11B1 (0.33) IDO1HSD11B1NOTUMNR1H2NR1H3
SCHEMBL1052795 0.77 HSD11B1 (0.42) IDO1HSD11B1ALDH1A1NOTUMCYP1A2
SCHEMBL29913869 0.73 ALDH1A1 (0.39) IDO1HSD11B1ALDH1A1NOTUMCYP1A2
SCHEMBL8983836 0.71 TSHR (0.39) ALDH1A1CYP3A4TDP1TSHRHSD17B10
Bromide SCHEMBL19405537 0.71 HSD11B1 (0.38) IDO1HSD11B1ALDH1A1NOTUMCYP1A2
Bromide SCHEMBL19405666 0.71 HSD11B1 (0.42) HSD11B1ALDH1A1NOTUMCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL19405387 0.71 HSD11B1 (0.42) HSD11B1ALDH1A1NOTUMCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL19405518 0.71 HSD11B1 (0.38) HSD11B1ALDH1A1NOTUMCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed
EP-0710241-A1 NOVEL SILYLATED BENZYLAMINE DERIVATIVES, SALTS THEREOF, METHODS OF MANUFACTURE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PIERRE FABRE MEDICAMENT (FR) 1996-05-08 EP disclosed
WO-1995003313-A1 NOVEL SILYLATED BENZYLAMINE DERIVATIVES, SALTS THEREOF, METHODS OF MANUFACTURE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PIERRE FABRE MEDICAMENT (FR) 1995-02-02 WO disclosed