SCHEMBL7521691

SCHEMBL7521691

CC[Si](CC)(CC)CSc1cc(C(C)(C)C)c(OC(C)=O)cc1C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.36
NR1H4 Q96RI1 1/20 0.33
KDM4E B2RXH2 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
PKM P14618 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
CFD P00746 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7522610 0.90 PTGS2 (0.37) PTGS2NR1H4NPC1LMNAPKM
SCHEMBL7525030 0.86 PTGS2 (0.32) PTGS2NR1H4NPC1LMNAPKM
SCHEMBL7515293 0.78 PTGS2 (0.38) PTGS2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7529855 0.78 PTGS2 (0.40) PTGS2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7522271 0.77 PTGS2 (0.43) PTGS2
SCHEMBL7524510 0.76 ALOX15 (0.48) PTGS2KDM4EALDH1A1HPGDCYP2C19
SCHEMBL7517750 0.75 KDM4E (0.33) NR1H4KDM4EUSP2ALDH1A1HPGD
SCHEMBL7519659 0.74 ALOX15 (0.35)
SCHEMBL7515913 0.70 VCAM1 (0.43)
SCHEMBL7526616 0.69 VCAM1 (0.38) PTGS2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed