SCHEMBL7523406

SCHEMBL7523406

N#Cc1ccccc1S(=O)(=O)NC(=O)Nc1cc(Cl)ccc1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 18/20 0.54
GRIK2 Q13002 1/20 0.51
FBP1 P09467 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7469874 0.91 GRIK1 (0.51) GRIK1GRIK2
SCHEMBL7466216 0.86 P2RY12 (0.47) FBP1
SCHEMBL7465474 0.78 P2RY12 (0.47)
SCHEMBL7531464 0.75 GRIK1 (0.56) GRIK1
SCHEMBL7463645 0.73 GRIK1 (0.54) GRIK1
SCHEMBL7559587 0.72 GRIK1 (0.66) GRIK1
SCHEMBL7528058 0.71 FLT1 (0.61) GRIK1
SCHEMBL3957527 0.71 GRIK1 (1.00) GRIK1GRIK2
SCHEMBL7522905 0.70 GRIK1 (0.50) GRIK1
SCHEMBL3961542 0.69 GRIK1 (1.00) GRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
US-5814631-A CHYMASE INHIBITOR, CARDIVASCULAR SUNTORY LIMITED (JP) 1998-09-29 US disclosed
EP-0795548-A1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LIMITED (JP) 1997-09-17 EP disclosed