SCHEMBL7523969

SCHEMBL7523969

C[Si](C)(C)CCOc1ccc(CBr)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.38
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
HTT P42858 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
LTA4H P09960 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
APP P05067 2/20 0.36
LMNA P02545 2/20 0.36
HSD17B10 Q99714 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050696 0.87 TP53 (0.33) HRH3KEAP1NFE2L2HTTCYP1A2
SCHEMBL9705589 0.81 TRPA1 (0.43) HRH3KEAP1NFE2L2HTTCYP1A2
SCHEMBL9705573 0.79 KCNA3 (0.50) HRH3L3MBTL1
SCHEMBL4122924 0.78 L3MBTL1 (0.53) HTTCYP1A2CYP2C19LTA4HLMNA
SCHEMBL4487824 0.78 LTA4H (0.53) CYP1A2LTA4HCYP2D6
SCHEMBL9705568 0.77 KCNA3 (0.48)
SCHEMBL10614694 0.77 KCNA3 (0.48)
SCHEMBL4086993 0.77 TRPA1 (0.40) HRH3KEAP1NFE2L2HTTCYP1A2
SCHEMBL9539656 0.77 KCNA3 (0.48)
SCHEMBL9829763 0.76 ACACB (0.42) HRH3KEAP1NFE2L2APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690066-B1 Phosphinic acid derivatives, their preparation as well as their use AVENTIS PHARMA GMBH (DE) 2002-03-13 EP disclosed
US-5707979-A INHIBITORS OF RETROVIRAL PROTEASE INHIBITORS FOR TREATMENT OF HIV HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-13 US disclosed
EP-0690066-A1 Phosphinic acid derivatives, their preparation as well as their use HOECHST AKTIENGESELLSCHAFT (DE) 1996-01-03 EP disclosed