SCHEMBL752503

SCHEMBL752503

Cc1ccc(S(=O)(=O)N2CCN(C(=O)COc3cccc(Cl)c3)CC2)cc1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PKM P14618 8/20 0.69
LMNA P02545 1/20 0.67
GAA P10253 6/20 0.66
ALDH1A1 P00352 2/20 0.63
SMN1; SMN2 Q16637 1/20 0.63
FKBP1A P62942 1/20 0.58
TDP1 Q9NUW8 1/20 0.55
ENPP2 Q13822 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7894190 0.89 PKM (0.76) PKMLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL752501 0.87 LMNA (0.88) PKMLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL752279 0.87 GAA (0.85) PKMLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL7890108 0.82 LMNA (0.79) PKMLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL10143924 0.80 PKM (0.62) PKMLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL9950592 0.80 GAA (0.67) PKMLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL15134821 0.79 GAA (0.74) GAAALDH1A1FKBP1ATDP1ENPP2
SCHEMBL9951161 0.79 PKM (0.71) PKMLMNAGAAALDH1A1SMN1; SMN2
SCHEMBL752687 0.78 NPC1 (0.67) PKMGAAALDH1A1
SCHEMBL9950690 0.78 PKM (0.83) PKMLMNAGAAALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016034742-A1 METHODS OF DIAGNOSING AND TREATING CANCER INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2016-03-10 WO disclosed
US-8138190-B2 Diaza heterocyclic amide compounds and their uses AMGEN INC. (US) 2012-03-20 US disclosed
US-8138190-B2 Diaza heterocyclic amide compounds and their uses AMGEN INC. (US) 2012-03-20 US disclosed
US-20090176768-A1 DIAZA HETEROCYCLIC AMIDE COMPOUNDS AND THEIR USES AMGEN INC. 2009-07-09 US disclosed
US-20090176768-A1 DIAZA HETEROCYCLIC AMIDE COMPOUNDS AND THEIR USES AMGEN INC. 2009-07-09 US disclosed
US-7524848-B2 Diaza heterocyclic amide compounds and their uses AMGEN INC. (US) 2009-04-28 US disclosed
US-7524848-B2 Diaza heterocyclic amide compounds and their uses AMGEN INC. (US) 2009-04-28 US disclosed
US-20070249626-A1 Diaza heterocyclic amide compounds and their uses AMGEN INC. 2007-10-25 US disclosed
US-20070249626-A1 Diaza heterocyclic amide compounds and their uses AMGEN INC. 2007-10-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176768-A1 DIAZA HETEROCYCLIC AMIDE COMPOUNDS AND THEIR USES GPR119, GLP1R, INSR PKM 1084/4885LMNA 2505/4885GAA 517/4885
US-20070249626-A1 Diaza heterocyclic amide compounds and their uses GPR119, GLP1R, INSR PKM 1084/4885LMNA 2505/4885GAA 517/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.