SCHEMBL7526797

SCHEMBL7526797

O=CNc1c(F)cccc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.44
SLC22A12 Q96S37 3/20 0.38
KIF11 P52732 1/20 0.38
ALDH1A1 P00352 3/20 0.35
CTSS P25774 2/20 0.35
PTGES2 Q9H7Z7 1/20 0.35
JAK2 O60674 1/20 0.34
NFE2L2 Q16236 2/20 0.33
KAT6A Q92794 1/20 0.33
TRPA1 O75762 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
HSD11B1 P28845 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11616035 0.88 ALDH1A1 (0.38) PTGS2ALDH1A1CTSSLMNAGAA
SCHEMBL423087 0.82 ALDH1A1 (0.42) ALDH1A1NFE2L2
SCHEMBL11614677 0.80 PTGS2 (0.46) PTGS2SLC22A12ALDH1A1CTSS
SCHEMBL883519 0.75 PTGS2 (0.44) PTGS2SLC22A12KIF11ALDH1A1JAK2
SCHEMBL7527600 0.74 EPHX2 (0.44) PTGS2SLC22A12ALDH1A1CTSSKAT6A
SCHEMBL7526792 0.74 PTGS2 (0.44) PTGS2SLC22A12ALDH1A1PTGES2JAK2
SCHEMBL21461560 0.73 GAA (0.45) PTGS2ALDH1A1LMNAGAA
SCHEMBL21186770 0.73 ERN1 (0.42) ALDH1A1
SCHEMBL16240458 0.73 ALDH1A1 (0.37) ALDH1A1LMNAGAA
Hydrochloric Acid SCHEMBL2771576 0.73 ALDH1A1 (0.52) PTGS2SLC22A12ALDH1A1PTGES2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP claimed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO claimed
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed
US-4125620-A HYPOTENSIVE BOEHRINGER INGELHEIM GMBH (DE) 1978-11-14 US disclosed