SCHEMBL7526973

SCHEMBL7526973

O=CNc1ccc(Br)cc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.39
OPRM1 P35372 1/20 0.37
APP P05067 1/20 0.35
MPO P05164 1/20 0.35
KDM5A P29375 1/20 0.34
HCAR1 Q9BXC0 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
RAB9A P51151 3/20 0.33
NPC1 O15118 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
FFAR1 O14842 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7530896 0.80 IDO1 (0.39) APPMPOKDM5ARXFP1RAB9A
SCHEMBL14433830 0.79 APP (0.35) APPKDM5ARXFP1RAB9AALDH1A1
SCHEMBL7527171 0.79 RAB9A (0.54) RAB9ANPC1ALDH1A1MAPTSMN1; SMN2
SCHEMBL28158377 0.76 APP (0.47) KDM1AOPRM1APPMPOHCAR1
SCHEMBL11942146 0.76 ALDH1A1 (0.52) KDM1AOPRM1MPOHCAR1RAB9A
SCHEMBL5434561 0.76 NPC1 (0.53) RAB9ANPC1ALDH1A1MAPTSMN1; SMN2
SCHEMBL7526970 0.75 KDM1A (0.39) KDM1AOPRM1APPMPOHCAR1
SCHEMBL38659023 0.75 KDM1A (0.39) KDM1AOPRM1MPOHCAR1RAB9A
SCHEMBL10465699 0.75 HSP90AA1 (0.41) KDM5ARAB9ANPC1ALDH1A1MAPT
SCHEMBL15001572 0.73 SLC22A12 (0.42) KDM1AOPRM1FFAR1FFAR4SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP claimed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO claimed
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed