SCHEMBL7530896

SCHEMBL7530896

O=CNc1ccc(F)cc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.39
PTGES2 Q9H7Z7 3/20 0.36
ALOX15 P16050 1/20 0.36
APP P05067 1/20 0.36
KDM5A P29375 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
KIF11 P52732 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
RAB9A P51151 1/20 0.34
IDH2 P48735 1/20 0.34
MPO P05164 1/20 0.33
ARNT P27540 1/20 0.33
EPAS1 Q99814 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28188269 0.81 TAS2R14 (0.47) RXFP1CYP2C19RAB9AMPOALDH1A1
SCHEMBL7526973 0.80 KDM1A (0.39) APPKDM5ARXFP1CYP1A2CYP2D6
SCHEMBL14433830 0.80 APP (0.35) APPKDM5ARXFP1KIF11CYP1A2
SCHEMBL7527171 0.80 RAB9A (0.54) CYP1A2CYP2D6CYP2C19RAB9AALDH1A1
SCHEMBL988638 0.76 ALDH1A1 (0.47) CYP2C19RAB9AMEN1ALDH1A1LMNA
SCHEMBL2096095 0.75 POLB (0.53) RXFP1CYP1A2CYP2D6CYP2C19RAB9A
SCHEMBL11404013 0.75 IDO1 (0.42) IDO1ALOX15APPCYP1A2CYP2D6
SCHEMBL22838141 0.75 IDO1 (0.42) IDO1PTGES2ALOX15CYP1A2CYP2D6
SCHEMBL15110952 0.75 ALDH1A1 (0.53) IDO1PTGES2ALOX15CYP1A2CYP2D6
SCHEMBL9229437 0.75 APP (0.49) IDO1PTGES2ALOX15APPKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP claimed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO claimed
EP-2888229-B1 alpha7 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS AND USES THEREOF MERCK SHARP & DOHME (US) 2019-02-06 EP disclosed
WO-2015192282-A1 FORMYLATION PROCESS FOR PREPARING AROMATIC FORMAMIDES RHODIA OPERATIONS (FR) 2015-12-23 WO disclosed
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed