SCHEMBL7527156

SCHEMBL7527156

[NH]C(=O)c1ccc(CBr)c([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 2/20 0.49
CASP6 P55212 1/20 0.45
CYP1A2 P05177 1/20 0.43
VCAM1 P19320 1/20 0.42
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
PARP1 P09874 1/20 0.41
GSK3B P49841 1/20 0.40
HCAR3 P49019 6/20 0.40
APEX1 P27695 1/20 0.39
SNCA P37840 1/20 0.39
PRSS1 P07477 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL40979 0.85 CASP6 (0.64) PDK1CASP6LMNATSHRHCAR3
SCHEMBL7510384 0.84 PARP1 (0.59) PDK1CASP6LMNATSHRPARP1
SCHEMBL28269442 0.84 PDK1 (0.52) PDK1CASP6CYP1A2VCAM1LMNA
SCHEMBL1018568 0.80 VCAM1 (0.58) PDK1VCAM1LMNA
SCHEMBL11321021 0.80 PDK1 (0.49) PDK1CYP1A2LMNATSHRHCAR3
SCHEMBL11321018 0.80 PDK1 (0.46) PDK1CASP6LMNAPARP1HCAR3
SCHEMBL13816452 0.78 PDK1 (0.50) PDK1CYP1A2LMNAHCAR3
SCHEMBL4262486 0.78 KMT2A (0.61) PDK1LMNA
SCHEMBL6953347 0.77 PDK1 (0.46) PDK1VCAM1LMNATSHR
Isothiocyanate SCHEMBL27833109 0.77 VCAM1 (0.54) PDK1CASP6VCAM1LMNAHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002020630-A1 PROCESS FOR THE PREPARATION OF GLYCEROL-BASED CROSSLINKED POLYMERIC GELS LIPAL BIOCHEMICALS (CH) 2002-03-14 WO disclosed