SCHEMBL7527652

SCHEMBL7527652

N=C(N)CCc1ccc(CCS(=O)(=O)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 6/20 0.45
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
F2 P00734 3/20 0.38
TMPRSS4 Q9NRS4 2/20 0.38
CYP2D6 P10635 2/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38
RECQL P46063 1/20 0.38
ALDH1A1 P00352 2/20 0.36
F10 P00742 1/20 0.36
LMNA P02545 1/20 0.36
NPC1 O15118 1/20 0.36
CYP3A4 P08684 1/20 0.36
NOS1 P29475 1/20 0.36
RAB9A P51151 1/20 0.36
HIF1A Q16665 1/20 0.36
BLM P54132 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7531044 0.82 PRSS1 (0.50) MGLLF2F10LMNAITGB3
SCHEMBL8780954 0.80 NOS1 (0.50) CA1CA2F2CYP2D6ALDH1A1
SCHEMBL4843038 0.75 IDO1 (0.53) CYP2D6NPC1CYP3A4NOS1RAB9A
SCHEMBL12401897 0.74 NOS1 (0.45) F2CYP2D6F10NPC1CYP3A4
Hydrochloric Acid SCHEMBL4714243 0.73 IDO1 (0.55) CYP2D6NPC1CYP3A4NOS1RAB9A
SCHEMBL12376924 0.72 NOS1 (0.43) F2CYP2D6F10NPC1CYP3A4
SCHEMBL12401872 0.72 CYP3A4 (0.43) CA2CYP2D6TP53ALDH1A1LMNA
SCHEMBL29001390 0.72 MGLL (0.48) MGLLCA1CA2F2TMPRSS4
SCHEMBL4847288 0.71 IDO1 (0.58) LMNA
SCHEMBL29001383 0.71 MGLL (0.47) MGLLCA1CA2CA12CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623146-B1 COMPOSITIONS AND METHODS FOR INHIBITING BETA-PROTEIN FUNCTION HARVARD COLLEGE (US) 2002-04-17 EP disclosed
US-5506097-A CONTACTING ALZHEIMER AMYLOID BETA-PROTEIN WITH EBELACTONE A OR PARA-AMIDINOPHENYLMETHANESULFONYL FLUORIDE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 1996-04-09 US disclosed
EP-0623146-A1 COMPOUNDS AND METHODS FOR INHIBITING $g(b)-PROTEIN FUNCTION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 1994-11-09 EP disclosed
WO-1993015112-A2 COMPOUNDS AND METHODS FOR INHIBITING β-PROTEIN FUNCTION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 1993-08-05 WO disclosed