SCHEMBL7529150

SCHEMBL7529150

CCCNc1cc(Cl)ccc1OC

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.55
MEN1 O00255 3/20 0.55
L3MBTL1 Q9Y468 2/20 0.54
NPSR1 Q6W5P4 2/20 0.54
ALDH1A1 P00352 5/20 0.51
POLB P06746 3/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C19 P33261 1/20 0.51
GAA P10253 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TP53 P04637 1/20 0.47
GBA1 P04062 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7527613 0.85 CYP1A2 (0.46) KMT2AMEN1L3MBTL1ALDH1A1POLB
SCHEMBL5663443 0.81 KMT2A (0.51) KMT2AMEN1L3MBTL1NPSR1ALDH1A1
SCHEMBL7531918 0.81 MAPT (0.59) KMT2AMEN1L3MBTL1ALDH1A1POLB
SCHEMBL11957889 0.81 KMT2A (0.61) KMT2AMEN1NPSR1ALDH1A1POLB
SCHEMBL11935558 0.80 RAD52 (0.51) KMT2AMEN1ALDH1A1POLBCYP1A2
SCHEMBL7526020 0.79 SMN1; SMN2 (0.45) KMT2AMEN1L3MBTL1ALDH1A1GAA
SCHEMBL7529112 0.79 PTGS2 (0.44) KMT2AMEN1L3MBTL1ALDH1A1POLB
SCHEMBL10798749 0.79 MEN1 (0.55) KMT2AMEN1L3MBTL1NPSR1ALDH1A1
SCHEMBL7535112 0.78 POLB (0.47) KMT2AMEN1L3MBTL1POLBGAA
SCHEMBL23565733 0.77 KMT2A (0.61) KMT2AMEN1NPSR1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020137740-A1 Aminothiazole derivatives, process for preparing them and pharmaceutical compositions containing them FONTAINE EVELYNE (FR) 2002-09-26 US disclosed
EP-0934290-B1 AMINOTHIAZOLE DERIVATIVES, METHOD OF PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI SYNTHELABO (FR) 2002-04-17 EP disclosed
US-6344470-B1 Aminothiazole derivatives, method of preparation and pharmaceutical compositions containing same SANOFI-SYNTHELABO (FR) 2002-02-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137740-A1 Aminothiazole derivatives, process for preparing them and pharmaceutical compositions containing them CRHR1, ADRA1D, ADRB1 KMT2A 2618/4885MEN1 2208/4885L3MBTL1 4761/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.