SCHEMBL7530810

SCHEMBL7530810

COC(=O)c1ccc(C)c(NC(=O)c2sccc2NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.58
CYP2C9 P11712 6/20 0.58
TSHR P16473 4/20 0.58
NPSR1 Q6W5P4 1/20 0.58
HPGD P15428 4/20 0.52
LMNA P02545 3/20 0.52
KMT2A Q03164 4/20 0.50
MEN1 O00255 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
KDM4E B2RXH2 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CRHBP P24387 1/20 0.50
CYP2C19 P33261 1/20 0.50
HTT P42858 1/20 0.50
CRHR2 Q13324 1/20 0.50
NOD2 Q9HC29 1/20 0.50
PKM P14618 1/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7534382 0.97 CYP2C9 (0.55) ALDH1A1CYP2C9TSHRNPSR1HPGD
SCHEMBL7532088 0.89 CYP2C9 (0.60) ALDH1A1CYP2C9TSHRNPSR1HPGD
SCHEMBL7537945 0.85 HPGD (0.67) ALDH1A1CYP2C9TSHRNPSR1HPGD
SCHEMBL7533940 0.84 RAB9A (0.56) ALDH1A1CYP2C9TSHRHPGDLMNA
SCHEMBL17331324 0.83 CYP2C9 (0.80) ALDH1A1CYP2C9TSHRNPSR1HPGD
SCHEMBL7530812 0.83 CYP2C9 (0.52) ALDH1A1CYP2C9TSHRNPSR1HPGD
SCHEMBL7530805 0.81 CYP2C9 (0.50) ALDH1A1CYP2C9TSHRNPSR1HPGD
SCHEMBL532885 0.80 LMNA (0.78) ALDH1A1CYP2C9TSHRNPSR1HPGD
SCHEMBL7531858 0.78 KMT2A (0.55) ALDH1A1TSHRHPGDLMNAKMT2A
SCHEMBL533542 0.78 FFAR4 (0.57) TSHRHPGDLMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002028353-A2 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-11 WO disclosed