SCHEMBL7531990

SCHEMBL7531990

COc1ccc(C(=O)NC2(C(=O)NCCCCC(=O)c3nc4ccccc4o3)CCCCC2)cc1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
LMNA P02545 2/20 0.42
TSHR P16473 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 3/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
LPAR1 Q92633 1/20 0.42
FAAH O00519 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7535950 0.85 CTSL (0.49) MAPTHDAC3HDAC4HDAC1HDAC7
SCHEMBL7533012 0.84 FAAH (0.45) POLBHDAC6FAAHCES1DAGLA
SCHEMBL7530297 0.84 CTSL (0.42) POLBHDAC3HDAC1HDAC6FAAH
SCHEMBL7529866 0.84 FAAH (0.43) POLBHDAC6FAAHCES1DAGLA
SCHEMBL7535321 0.84 FAAH (0.43) POLBHDAC3HDAC1HDAC6FAAH
SCHEMBL7537229 0.82 HDAC3 (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7536597 0.82 FAAH (0.43) ALDH1A1LMNAPOLBNPC1RAB9A
SCHEMBL7531275 0.82 TACR2 (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7532252 0.81 CTSL (0.54) ALDH1A1MAPTHDAC3HDAC1NPC1
SCHEMBL7528076 0.81 CTSL (0.54) ALDH1A1LMNATSHRNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002023784-A2 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-03-21 WO disclosed