SCHEMBL7533428

SCHEMBL7533428

CCCCOC(=O)N1CCC(C(=O)O)CC1.CCCCOC(=O)N1CCC(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.70
NPC1 O15118 3/20 0.70
RAB9A P51151 3/20 0.70
CYP2C19 P33261 1/20 0.57
HTT P42858 1/20 0.52
MAPT P10636 1/20 0.50
ALDH1A1 P00352 2/20 0.48
TSHR P16473 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
CYP3A4 P08684 1/20 0.48
MAPK1 P28482 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
POLB P06746 2/20 0.46
S1PR5 Q9H228 1/20 0.46
NPSR1 Q6W5P4 2/20 0.45
ENPP2 Q13822 1/20 0.45
LTA4H P09960 1/20 0.45
KDM4E B2RXH2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6999819 0.97 NPC1 (0.63) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL10408085 0.88 SMN1; SMN2 (0.64) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL6178689 0.85 NPC1 (0.60) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL7299227 0.83 L3MBTL1 (0.59) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL2175396 0.83 TSHR (0.59) MAPTALDH1A1TSHRL3MBTL1CYP3A4
SCHEMBL205216 0.83 SMN1; SMN2 (1.00) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL355693 0.83 SMN1; SMN2 (0.58) SMN1; SMN2NPC1RAB9AHTTMAPT
SCHEMBL630697 0.82 SMN1; SMN2 (0.73) SMN1; SMN2NPC1RAB9ACYP2C19HTT
Hydrochloric Acid SCHEMBL3097843 0.82 SMN1; SMN2 (0.97) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL3664936 0.80 LMNA (0.58) SMN1; SMN2NPC1RAB9ACYP2C19HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165540-A1 TETRAHYDROPYRAN DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 2002-01-02 EP disclosed
WO-2000056727-A1 TETRAHYDROPYRAN DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 2000-09-28 WO disclosed
WO-2000056728-A1 TETRAHYDROPYRAN DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 2000-09-28 WO disclosed