SCHEMBL7534115

SCHEMBL7534115

CC(C)c1ccc(-n2nc(-c3cccs3)c3c2C(=O)CCC3(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
DHODH Q02127 1/20 0.35
ALDH1A1 P00352 5/20 0.34
HSD17B10 Q99714 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALPL P05186 1/20 0.34
HPGD P15428 1/20 0.34
MAPT P10636 4/20 0.33
KDM5B Q9UGL1 1/20 0.32
TP53 P04637 2/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
PARP1 P09874 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
TRPV4 Q9HBA0 1/20 0.32
NPC1 O15118 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
EGFR P00533 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7537152 0.83 DHODH (0.40) DHODHALDH1A1KDM4EHPGDMAPT
SCHEMBL7533976 0.81 PARP1 (0.33) DHODHALDH1A1HPGDMAPTSMN1; SMN2
SCHEMBL7483421 0.80 DHODH (0.43) DHODHMAPTKDM5BTRPV4CYP1A2
SCHEMBL7488250 0.80 PTGS1 (0.45) POLBDHODHALDH1A1HSD17B10KDM4E
SCHEMBL7484570 0.78 GAA (0.35) DHODHMAPTKDM5BGAA
SCHEMBL7537246 0.77 DHODH (0.41) DHODHMAPTKDM5BRAB9ANPSR1
SCHEMBL7534112 0.75 OPRM1 (0.50) POLBALDH1A1HSD17B10KDM4EALPL
SCHEMBL6767179 0.67 POLB (0.35) POLBDHODHALDH1A1HSD17B10KDM4E
SCHEMBL6164575 0.65 CCNA2 (0.38) ALDH1A1HSD17B10KDM4EALPLHPGD
SCHEMBL6770073 0.65 MAPT (0.34) DHODHALDH1A1MAPTSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed