SCHEMBL7534112

SCHEMBL7534112

CC(C)c1ccc(-n2nc(-c3cccs3)c3c2CC(C)(C)CC3=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 14/20 0.50
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALPL P05186 1/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
SRC P12931 2/20 0.41
HSP90AB1 P08238 1/20 0.38
OPRD1 P41143 2/20 0.38
OPRK1 P41145 2/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7537151 0.84 OPRM1 (0.54) OPRM1ALDH1A1HSD17B10SRC
SCHEMBL7533974 0.82 OPRM1 (0.47) OPRM1ALDH1A1SRCHSP90AB1
SCHEMBL6767179 0.81 POLB (0.35) OPRM1ALDH1A1KDM4EALPLHPGD
SCHEMBL7483415 0.80 OPRM1 (0.49) OPRM1SRCHSP90AB1OPRD1OPRK1
SCHEMBL7488247 0.80 OPRM1 (0.49) OPRM1SRCHSP90AB1OPRD1OPRK1
SCHEMBL6767006 0.79 OPRM1 (0.58) OPRM1SRCHSP90AB1OPRD1OPRK1
SCHEMBL6770401 0.79 OPRM1 (0.77) OPRM1ALDH1A1HSD17B10HSP90AB1OPRD1
SCHEMBL7484568 0.79 OPRM1 (0.50) OPRM1SRCHSP90AB1OPRD1OPRK1
SCHEMBL7479730 0.78 OPRM1 (0.54) OPRM1ALDH1A1SRCHSP90AB1OPRD1
SCHEMBL7537240 0.78 OPRM1 (0.58) OPRM1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed