SCHEMBL7537152

SCHEMBL7537152

CC(C)c1ccc(-n2nc(-c3ccccc3)c3c2C(=O)CCC3(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.40
SRC P12931 2/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
ALDH1A1 P00352 5/20 0.34
PTGS2 P35354 3/20 0.34
PTGS1 P23219 2/20 0.34
MEN1 O00255 5/20 0.34
KMT2A Q03164 5/20 0.34
HTT P42858 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 2/20 0.33
NPBWR1 P48145 1/20 0.33
MCHR1 Q99705 1/20 0.33
PIK3CD O00329 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7484570 0.87 GAA (0.35) DHODHSRCPTGS2PTGS1MAPT
SCHEMBL7537246 0.87 DHODH (0.41) DHODHSRCCA1CA2RAB9A
SCHEMBL7483421 0.86 DHODH (0.43) DHODHMAPTPIK3CDPIK3R2PIK3CA
SCHEMBL7488250 0.83 PTGS1 (0.45) DHODHALDH1A1PTGS1MEN1KMT2A
SCHEMBL7534115 0.83 POLB (0.36) DHODHALDH1A1MEN1KMT2AHTT
SCHEMBL7533976 0.74 PARP1 (0.33) DHODHALDH1A1MEN1KMT2AHTT
SCHEMBL7537151 0.73 OPRM1 (0.54) SRCALDH1A1MEN1KMT2AHTT
SCHEMBL6772430 0.68 CCNA2 (0.44) DHODHSRCALDH1A1MEN1KMT2A
SCHEMBL5214539 0.67 KMT2A (0.49) DHODHSRCCA1CA2ALDH1A1
SCHEMBL6770531 0.65 MEN1 (0.40) DHODHSRCALDH1A1PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed