SCHEMBL7537246

SCHEMBL7537246

COc1cccc(-c2nn(-c3ccc(C(C)C)cc3)c3c2C(C)(C)CCC3=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.41
SRC P12931 3/20 0.40
DGAT2 Q96PD7 1/20 0.37
NPBWR1 P48145 5/20 0.37
MCHR1 Q99705 4/20 0.37
ROCK2 O75116 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
LMNA P02545 2/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
SLC16A3 O15427 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7537152 0.87 DHODH (0.40) DHODHSRCNPBWR1MCHR1LMNA
SCHEMBL7484570 0.79 GAA (0.35) DHODHSRCNPBWR1MCHR1KDM5B
SCHEMBL7488250 0.79 PTGS1 (0.45) DHODHMAPTTSHRNPSR1
SCHEMBL7483421 0.78 DHODH (0.43) DHODHKDM5BMAPT
SCHEMBL7537240 0.78 OPRM1 (0.58) DHODHSRCMAPTCA1CA2
SCHEMBL7534115 0.77 POLB (0.36) DHODHKDM5BMAPTRAB9ANPSR1
SCHEMBL6772794 0.73 CCNA2 (0.40) DHODHSRCDGAT2NPBWR1MCHR1
SCHEMBL6777360 0.71 OPRM1 (0.39) DHODHSRCDGAT2NPBWR1MCHR1
SCHEMBL7533976 0.69 PARP1 (0.33) DHODHLMNAMAPTTSHRNPSR1
SCHEMBL6166539 0.69 SRC (0.39) DHODHSRCMAPTRAB9ASLC16A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed