SCHEMBL7535840

SCHEMBL7535840

COc1c(C)c[nH]c(=O)c1-c1ccc(C[C@H](N)C(=O)O)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 7/20 0.43
SLC7A5 Q01650 2/20 0.43
ALPI P09923 1/20 0.41
PKM P14618 1/20 0.41
PTGS1 P23219 1/20 0.41
XIAP P98170 1/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
GPR142 Q7Z601 2/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
PTPRC P08575 1/20 0.39
PTPN1 P18031 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7533946 0.89 ALDH1A1 (0.42) TPH1PPARGPPARAGPR142
SCHEMBL7535596 0.74 ITGA4 (0.48) ITGB3ITGA2BPTPN1
SCHEMBL22189982 0.74 SLC7A5 (0.61) TPH1SLC7A5ALPIPKMPTGS1
SCHEMBL22189984 0.74 SLC7A5 (0.61) TPH1SLC7A5ALPIPKMPTGS1
SCHEMBL7227087 0.72 ITGB1 (0.56) TPH1SLC7A5ALPIPKMPTGS1
SCHEMBL5162726 0.72 ITGB1 (0.56) TPH1SLC7A5ALPIPKMPTGS1
Hydrochloric Acid SCHEMBL7419313 0.71 ALDH1A1 (0.42) TPH1PPARGPPARAGPR142
SCHEMBL7416021 0.71 GPR142 (0.40) PPARGPPARAGPR142
SCHEMBL6168594 0.71 TPH1 (0.68) TPH1SLC7A5ALPIPKMPTGS1
Hydrochloric Acid SCHEMBL5159881 0.71 ITGB1 (0.55) TPH1SLC7A5ALPIPKMPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002008202-A2 ALPHA AMINO ACID DERIVATIVES--INHIBITORS OF LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2002-01-31 WO disclosed