SCHEMBL7536657

SCHEMBL7536657

CCCOCc1nc2nc(N(O)O)[nH]c(=O)c2[nH]1

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 11/20 0.33
PNP P00491 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10421279 0.79 PNP (0.54) PNP
SCHEMBL7536668 0.72 PDE5A (0.36)
SCHEMBL37957 0.69 PNP (0.53) PNP
SCHEMBL1767745 0.69 PNP (0.56) PNP
SCHEMBL4730342 0.69 FGFR1 (0.34) PNP
SCHEMBL17437739 0.67 ADORA3 (0.33)
SCHEMBL9191469 0.65 HCAR2 (0.47) HCAR2
SCHEMBL8397615 0.64 PNP (0.54) PNP
SCHEMBL16028668 0.63 POLB (0.68)
SCHEMBL2343355 0.62 PNP (0.59) PNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0684822-B1 CARBOCYCLIC DEOXYGUANOSINE ANALOGS FOR THE TREATMENT OF VIRAL INFECTIONS SOUTHERN RES INST (US) 2002-05-08 EP disclosed
US-6080746-A ADMINISTERING PURINE DERIVATIVE FOR PROPHYLAXIS AND TREATMENT OF CYTOMEGALO VIURS INFECTIONS IN HUMANS SOUTHERN RESEARCH INSTITUTE 2000-06-27 US disclosed
US-6001840-A A SUBSTANTIAL MOLAR EXCESS OF THE D-STEREOISOMER OF 2'CDG OVER THE L-STEREOISOMER. SOUTHERN RESEARCH INSTITUTE (US) 1999-12-14 US disclosed
US-5718922-A Intravitreal microsphere drug delivery and method of preparation SCHEPENS EYE RESEARCH INSTITUTE, INC. (US) 1998-02-17 US disclosed
WO-1996038133-A1 INTRAVITREAL MICROSPHERE DRUG DELIVERY AND METHOD OF PREPARATION SCHEPENS EYE RESEARCH INSTITUTE, INC. (US) 1996-12-05 WO disclosed
EP-0684822-A4 1996-01-10 EP disclosed
EP-0684822-A1 METHODS OF TREATMENT OF VIRAL INFECTIONS USING CARBOCYCLIC DEOXYGUANOSINE ANALOGS SOUTHERN RESEARCH INSTITUTE (US) 1995-12-06 EP disclosed
WO-1994018979-A2 METHODS OF TREATMENT OF VIRAL INFECTIONS USING CARBOCYCLIC DEOXYGUANOSINE ANALOGS SOUTHERN RESEARCH INSTITUTE (US) 1994-09-01 WO disclosed
EP-0471057-A4 METHODS AND COMPOSITIONS FOR THE PROPHYLAXIS AND TREATMENT OF CYTOMEGALOVIRUS INFECTIONS 1992-11-19 EP disclosed
EP-0471057-A1 METHODS AND COMPOSITIONS FOR THE PROPHYLAXIS AND TREATMENT OF CYTOMEGALOVIRUS INFECTIONS VIRACHEM, INC. (US) 1992-02-19 EP disclosed
WO-1991013549-A1 METHODS AND COMPOSITIONS FOR THE PROPHYLAXIS AND TREATMENT OF CYTOMEGALOVIRUS INFECTIONS VIRACHEM, INC. (US) 1991-09-19 WO disclosed
US-4849412-A PAPAVERINE COMPOUND, NUCLEOSIDE ANALOG BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1989-07-18 US disclosed
WO-1987007508-A1 METHODS AND COMPOSITIONS FOR TREATING VIRAL INFECTIONS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1987-12-17 WO disclosed