SCHEMBL7538682

SCHEMBL7538682

COC(=O)[C@H](Cc1ccc(OCC(C)C)cc1)NC(=O)[C@@H](OCc1ccc2ccccc2c1)C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
TSHR P16473 1/20 0.46
PPARG P37231 3/20 0.45
PPARD Q03181 2/20 0.45
PPARA Q07869 2/20 0.45
HDAC1 Q13547 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
ADAM17 P78536 1/20 0.43
THRB P10828 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
IL1RN P18510 2/20 0.42
ERAP2 Q6P179 2/20 0.42
ERAP1 Q9NZ08 2/20 0.42
MAOB P27338 1/20 0.42
TACR1 P25103 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7538679 1.00 ALDH1A1 (0.46) ALDH1A1MEN1LMNAKMT2ATSHR
SCHEMBL7539918 0.92 MME (0.50) PPARGADAM17MAOB
SCHEMBL7543915 0.92 MME (0.50) PPARGADAM17MAOB
SCHEMBL7541085 0.80 ALDH1A1 (0.53) ALDH1A1MEN1LMNAKMT2ATSHR
SCHEMBL7541086 0.80 ALDH1A1 (0.53) ALDH1A1MEN1LMNAKMT2ATSHR
SCHEMBL7538549 0.75 YAP1 (0.51) ALDH1A1MEN1LMNAKMT2ATSHR
SCHEMBL7538553 0.75 YAP1 (0.51) ALDH1A1MEN1LMNAKMT2ATSHR
SCHEMBL27564126 0.73 ITGB3 (0.55) ALDH1A1MEN1LMNAKMT2AGAA
SCHEMBL7540882 0.72 MME (0.55) PPARG
SCHEMBL7540879 0.72 MME (0.55) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1209147-A1 CARBOXYLIC ACID DERIVATIVES AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2002-05-29 EP disclosed