SCHEMBL7538698

SCHEMBL7538698

N=C1CCCN1c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.56
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
ALOX5 P09917 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
INMT O95050 2/20 0.38
POLB P06746 1/20 0.38
SCN1A P35498 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3864473 0.81 ALDH1A1 (0.45) SIGMAR1MEN1NPC1RAB9AKMT2A
Hydrochloric Acid SCHEMBL5631058 0.79 ALDH1A1 (0.48) SIGMAR1MEN1NPC1RAB9AKMT2A
Hydrochloric Acid SCHEMBL11721493 0.78 RAB9A (0.43) SIGMAR1RAB9AALOX5KDM4EALDH1A1
Hydrochloric Acid SCHEMBL6771290 0.77 ALDH1A1 (0.65) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL14199843 0.77 SIGMAR1 (0.82) SIGMAR1MEN1NPC1RAB9AKMT2A
SCHEMBL4426213 0.76 SIGMAR1 (0.46) SIGMAR1MEN1NPC1RAB9AKMT2A
SCHEMBL6140774 0.75 KMT2A (0.43) MEN1NPC1RAB9AKMT2AALDH1A1
SCHEMBL3868815 0.75 ALDH1A1 (0.48) SIGMAR1MEN1NPC1RAB9AKMT2A
SCHEMBL21507867 0.74 SIGMAR1 (0.45) SIGMAR1MEN1NPC1RAB9AKMT2A
SCHEMBL29052583 0.74 SIGMAR1 (0.45) SIGMAR1MEN1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934265-A1 AMIDINOPHENYL-PYRROLIDINES, -PYRROLINES, AND -ISOXAZOLIDINES AND DERIVATIVES THEREOF Du Pont Pharmaceuticals Company (US) 1999-08-11 EP disclosed
WO-1998006694-A1 AMIDINOPHENYL-PYRROLIDINES, -PYRROLINES, AND -ISOXAZOLIDINES AND DERIVATIVES THEREOF DU PONT PHARMACEUTICALS COMPANY (US) 1998-02-19 WO disclosed
US-4052382-A 1-PHENYL-3-AZACARBOCYCLIC-UREAS STERLING DRUG INC. (US) 1977-10-04 US disclosed
US-4026938-A 1-Phenyl-3-azacarbocyclic-ureas STERLING DRUG INC. (US) 1977-05-31 US disclosed
US-3963748-A 1-Phenyl-3-azacarbocyclic-ureas STERLING DRUG INC. (US) 1976-06-15 US disclosed