SCHEMBL753879

SCHEMBL753879

O=C(O)NC1C2CN(c3ccc(-c4ccc(F)cc4)cn3)CC21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.41
DRD4 P21917 2/20 0.41
HTR2A P28223 2/20 0.41
SLC6A4 P31645 2/20 0.41
DRD3 P35462 2/20 0.41
ACACB O00763 1/20 0.41
KCNH2 Q12809 2/20 0.40
DGAT1 O75907 1/20 0.40
ADORA2A P29274 1/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC3 O15379 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762021 0.85 RAB9A (0.40) ACACBKCNH2DGAT1ADORA2AHDAC2
SCHEMBL1729788 0.81 TDO2 (0.53) HTR1ADRD4HTR2ASLC6A4DRD3
SCHEMBL3722907 0.78 DGAT1 (0.40) HTR1ADRD4HTR2ASLC6A4DRD3
SCHEMBL3719971 0.76 DGAT1 (0.43) HTR1ADRD4HTR2ASLC6A4DRD3
SCHEMBL16174434 0.76 GRM1 (0.43) HTR1ADRD4HTR2ASLC6A4DRD3
SCHEMBL16174433 0.76 GRM1 (0.43) HTR1ADRD4HTR2ASLC6A4DRD3
SCHEMBL3477140 0.76 HDAC3 (0.47) HTR1AACACBHDAC2HDAC3HDAC1
SCHEMBL15653977 0.75 DGAT1 (0.40) HTR1ADRD4HTR2ASLC6A4DRD3
SCHEMBL14796957 0.74 CKS1B (0.48) HTR1ADRD4HTR2ASLC6A4DRD3
SCHEMBL8512363 0.74 KMT2A (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429998-A1 5-MEMBERED HETEROCYCLIC COMPOUND CYCLOPENTA[C]PYRROLYLALKYLCARBAMATE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-21 EP claimed
WO-2010130943-A1 5-MEMBERED HETEROCYCLIC COMPOUND CYCLOPENTA[C]PYRROLYLALKYLCARBAMATE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2010-11-18 WO claimed