SCHEMBL7539260

SCHEMBL7539260

CC(C)(C)COC(=O)NC(Cc1ccc2c(c1)Cc1cc(CCNc3nc4ccccc4[nH]3)ccc1-2)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.45
ITGA5 P08648 1/20 0.45
PTPN1 P18031 1/20 0.45
ITGB3 P05106 13/20 0.43
ITGAV P06756 13/20 0.43
BCHE P06276 1/20 0.43
PIN1 Q13526 3/20 0.42
ITGA2B P08514 1/20 0.39
ITGB5 P18084 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7540177 0.80 ITGAV (0.43) ITGB3ITGAVITGA2B
SCHEMBL7542370 0.79 BCHE (0.43) ITGB1ITGA5ITGB3ITGAVBCHE
SCHEMBL3048231 0.78 ITGB3 (0.45) ITGB1ITGA5PTPN1ITGB3ITGAV
SCHEMBL5204539 0.71 ITGB3 (0.41) ITGB1ITGA5PTPN1ITGB3ITGAV
SCHEMBL8657006 0.69 ACE (0.60) ITGB1PTPN1ITGB3ITGAVITGA2B
SCHEMBL11032508 0.69 ACE (0.60) ITGB1PTPN1ITGB3ITGAVITGA2B
SCHEMBL1712913 0.68 ACE (0.53) ITGB3ITGAVITGA2B
SCHEMBL1712911 0.68 ACE (0.53) ITGB3ITGAVITGA2B
SCHEMBL14431792 0.66 BCHE (0.37) ITGB1ITGA5ITGB3ITGAVBCHE
SCHEMBL31370428 0.65 PTPN1 (0.49) PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208088-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2002-05-29 EP disclosed
WO-2001010841-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2001-02-15 WO disclosed