SCHEMBL7540177

SCHEMBL7540177

CC(C)(C)COC(=O)NC(Cc1ccc2c(c1)Cc1cc(CCNC3=NCCN3)ccc1-2)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 18/20 0.43
ITGB3 P05106 18/20 0.43
ITGB6 P18564 1/20 0.38
MME P08473 1/20 0.37
ACE P12821 1/20 0.37
ITGA2B P08514 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13170299 0.82 ACE (0.46) ITGAVITGB3ITGB6MMEACE
SCHEMBL7539260 0.80 ITGB1 (0.45) ITGAVITGB3ITGA2B
SCHEMBL7241839 0.69 ITGB3 (0.51) ITGAVITGB3ITGA2B
SCHEMBL8657006 0.67 ACE (0.60) ITGAVITGB3MMEACEITGA2B
SCHEMBL11032508 0.67 ACE (0.60) ITGAVITGB3MMEACEITGA2B
SCHEMBL1712913 0.66 ACE (0.53) ITGAVITGB3MMEACEITGA2B
SCHEMBL1712911 0.66 ACE (0.53) ITGAVITGB3MMEACEITGA2B
SCHEMBL7242454 0.65 ITGB3 (0.57) ITGAVITGB3ITGA2B
SCHEMBL30171991 0.64 CXCR4 (0.45) ITGAVITGB3ITGB6ITGA2B
SCHEMBL14598327 0.63 CTSS (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208088-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2002-05-29 EP claimed
WO-2001010841-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2001-02-15 WO claimed
EP-1208088-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2002-05-29 EP disclosed
WO-2001010841-A2 FLUORENE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2001-02-15 WO disclosed