SCHEMBL753988

SCHEMBL753988

CN(C)CCCC(=O)NC1CC1.COc1ccc(Oc2ccc(CNC(=O)O)cc2)c(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
EPHX2 P34913 7/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SIRT1 Q96EB6 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
ALDH1A1 P00352 2/20 0.37
SLC6A5 Q9Y345 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL754465 0.84 AR (0.40) EPHX2SMN1; SMN2NPC1RAB9ASIGMAR1
SCHEMBL764430 0.82 SIRT1 (0.39) EPHX2SIRT1ALDH1A1
SCHEMBL755016 0.81 EPHX2 (0.46) EPHX2SMN1; SMN2ALDH1A1
Cyclopropane SCHEMBL3650772 0.81 EPHX2 (0.47) EPHX2PPARG
SCHEMBL10121383 0.79 SIRT1 (0.42) EPHX2SIRT1ALDH1A1
SCHEMBL13166418 0.78 POLB (0.42) EPHX2SIRT1KMT2A
SCHEMBL13165630 0.77 POLB (0.39) EPHX2SIRT1MEN1KMT2AALDH1A1
SCHEMBL10121546 0.76 L3MBTL1 (0.39) CYP2C19EPHX2MEN1KMT2AALDH1A1
SCHEMBL13165637 0.76 POLB (0.42) EPHX2SIRT1KMT2A
SCHEMBL756146 0.76 EPHX2 (0.61) EPHX2SMN1; SMN2NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed
EP-2188254-A1 NOVEL BRADYKININ B1-ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-05-26 EP disclosed
WO-2009027450-A1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-05 WO disclosed