SCHEMBL755016

SCHEMBL755016

COc1ccc(Oc2ccc(CNC(=O)O)cc2)c(C(F)(F)F)c1.NC1CC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 9/20 0.46
PTPN7 P35236 2/20 0.43
DUSP3 P51452 2/20 0.43
ALDH1A1 P00352 3/20 0.43
TSHR P16473 1/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclopropane SCHEMBL3650772 0.91 EPHX2 (0.47) EPHX2PTPN7DUSP3POLBL3MBTL1
SCHEMBL756146 0.85 EPHX2 (0.61) EPHX2ALDH1A1TSHRPOLBSMN1; SMN2
SCHEMBL754513 0.84 ALDH1A1 (0.48) ALDH1A1TSHRPOLBSMN1; SMN2
SCHEMBL754465 0.83 AR (0.40) EPHX2ALDH1A1TSHRSMN1; SMN2
SCHEMBL2549180 0.82 L3MBTL1 (0.45) EPHX2PTPN7DUSP3ALDH1A1POLB
SCHEMBL753988 0.81 CYP1A2 (0.41) EPHX2ALDH1A1SMN1; SMN2
SCHEMBL2787692 0.81 P2RX7 (0.42) EPHX2PTPN7DUSP3ALDH1A1POLB
SCHEMBL2542232 0.81 EPHX2 (0.44) EPHX2PTPN7DUSP3L3MBTL1
Trifluoroacetic Acid SCHEMBL2541472 0.81 HDAC3 (0.43) EPHX2PTPN7DUSP3L3MBTL1
SCHEMBL3642389 0.80 L3MBTL1 (0.43) EPHX2PTPN7DUSP3ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed