SCHEMBL7540238

SCHEMBL7540238

CC(C)C[C@H](NC(=O)c1ccc(-c2csc(N3CCN(C)CC3)n2)cc1)C(=O)N(C)C#N

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 14/20 0.58
CTSS P25774 13/20 0.57
CTSL P07711 11/20 0.57
CTSB P07858 9/20 0.53
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7486127 0.91 CTSK (0.55) CTSKCTSSCTSLCTSBNPC1
SCHEMBL6185770 0.90 CTSK (0.56) CTSKCTSSCTSLCTSB
SCHEMBL6182464 0.86 CTSK (0.64) CTSKCTSSCTSLCTSB
SCHEMBL6404499 0.85 CTSK (0.48) CTSKCTSSCTSLCTSBNPC1
SCHEMBL7450076 0.83 CTSB (0.54) CTSKCTSSCTSLCTSBNPC1
SCHEMBL7450318 0.83 CTSB (0.54) CTSKCTSSCTSLCTSB
SCHEMBL6185994 0.83 CTSB (0.54) CTSKCTSSCTSLCTSBNPC1
SCHEMBL6184402 0.83 CTSK (0.61) CTSKCTSSCTSLCTSB
SCHEMBL7507757 0.82 CTSK (0.54) CTSKCTSSCTSLCTSB
SCHEMBL6184317 0.81 CTSS (0.56) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO claimed