SCHEMBL7541979

SCHEMBL7541979

COCCOc1cc2oc(=O)cc(C)c2cc1C1=NCCN1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 5/20 0.39
KDM4E B2RXH2 10/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
ALDH1A1 P00352 8/20 0.39
HPGD P15428 7/20 0.39
HSD17B10 Q99714 7/20 0.39
GAA P10253 4/20 0.39
GLA P06280 3/20 0.39
CASP1 P29466 2/20 0.39
CASP7 P55210 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
MAPT P10636 1/20 0.39
ALPG P10696 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
ATM Q13315 2/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7537705 0.87 MAOB (0.39) ALDH1A1HSD17B10
SCHEMBL8218532 0.74 NISCH (0.38) KDM4E
SCHEMBL7543472 0.71 KDM4E (0.36) KDM4E
Hydrochloric Acid SCHEMBL8218663 0.71 KDM4E (0.39) KDM4E
SCHEMBL7485681 0.70 KDM4E (0.50) KDM4ECYP1A2CYP2C19ALDH1A1HPGD
SCHEMBL8198539 0.69 MC4R (0.49) GAASMN1; SMN2MAPT
SCHEMBL7536725 0.69 NISCH (0.32) KDM4E
Hydrochloric Acid SCHEMBL8203684 0.69 MC4R (0.46) KDM4ESMN1; SMN2MAPT
SCHEMBL9221587 0.68 KDM4E (0.56) KDM4ECYP1A2CYP2C19ALDH1A1HPGD
SCHEMBL6824821 0.68 MC4R (0.43) KDM4ESMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204644-A1 SYNTHESIS OF SUBSTITUTED AMIDINES ELI LILLY AND COMPANY (US) 2002-05-15 EP disclosed
WO-2000078725-A1 SYNTHESIS OF SUBSTITUTED AMIDINES ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed
WO-2000078724-A2 IMIDAZOLINDERIVATIVES THEIR PREPARATION AND THEIR PHARMACEUTICAL USE ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed