SCHEMBL7543472

SCHEMBL7543472

COCCOc1cc2c(cc1C1=NCCN1)CCCCC2

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
NISCH Q9Y2I1 8/20 0.35
HRH3 Q9Y5N1 1/20 0.34
PDCD1LG2 Q9BQ51 1/20 0.34
CD274 Q9NZQ7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8218663 0.97 KDM4E (0.39) KDM4EADRA2AADRA2BADRA2CNISCH
SCHEMBL8218198 0.87 NISCH (0.40) KDM4EADRA2AADRA2BADRA2CNISCH
Iodide SCHEMBL7537909 0.84 NOS3 (0.36) ADRA2AADRA2BADRA2CNISCHHRH3
SCHEMBL7538424 0.84 REN (0.33) KDM4EADRA2ANISCHPDCD1LG2CD274
Iodide SCHEMBL7537243 0.81 ESR1 (0.36) ADRA2AADRA2BADRA2CNISCHHRH3
SCHEMBL8218532 0.79 NISCH (0.38) KDM4EADRA2AADRA2BADRA2CNISCH
SCHEMBL8208937 0.78 PDCD1LG2 (0.35) KDM4ENISCHPDCD1LG2CD274
SCHEMBL7542447 0.78 KMT2A (0.42) KDM4E
SCHEMBL7536889 0.77 NISCH (0.36) KDM4EADRA2AADRA2BADRA2CNISCH
Iodide SCHEMBL7536945 0.76 POLB (0.40) KDM4EHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204644-A1 SYNTHESIS OF SUBSTITUTED AMIDINES ELI LILLY AND COMPANY (US) 2002-05-15 EP disclosed
WO-2000078725-A1 SYNTHESIS OF SUBSTITUTED AMIDINES ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed
WO-2000078724-A2 IMIDAZOLINDERIVATIVES THEIR PREPARATION AND THEIR PHARMACEUTICAL USE ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed