SCHEMBL7543655

SCHEMBL7543655

O=C(Cl)c1ccc(C(F)(F)F)cc1.O=C(Cl)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.50
CES1 P23141 2/20 0.50
TSHR P16473 1/20 0.48
SRD5A2 P31213 2/20 0.44
GSK3B P49841 2/20 0.43
PTPN1 P18031 1/20 0.43
KCNQ3 O43525 1/20 0.43
KCNQ2 O43526 1/20 0.43
KCNE1 P15382 1/20 0.43
KCNQ1 P51787 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.43
KMO O15229 2/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
RAD51 Q06609 1/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL68177 0.85 CES2 (0.67) CES2CES1TSHRSRD5A2GSK3B
SCHEMBL110094 0.83 TSHR (0.67) TSHRSRD5A2KCNQ3KCNQ2KCNE1
SCHEMBL29514652 0.83 TSHR (0.67) TSHRSRD5A2KCNQ3KCNQ2KCNE1
SCHEMBL2766866 0.80 SRD5A2 (0.68) CES2CES1TSHRSRD5A2GSK3B
SCHEMBL3992424 0.80 CES2 (0.59) CES2CES1TSHRSRD5A2GSK3B
SCHEMBL31542016 0.77 KDR (0.54) MEN1KMT2ALMNAMAPT
SCHEMBL1794695 0.77 KDR (0.54) MEN1KMT2ALMNAMAPT
SCHEMBL10532934 0.77 KMO (0.43) CES2TSHRKCNQ3KCNQ2KCNE1
SCHEMBL19970598 0.77 CES2 (0.55) CES2CES1TSHRSRD5A2GSK3B
SCHEMBL4254016 0.76 NPC1 (0.71) KCNQ3KCNQ2KCNE1KCNQ1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1064273-B1 1,3,4-THIADIAZOLES USEFUL FOR THE TREATMENT OF CMV INFECTIONS UPJOHN CO (US) 2002-12-18 EP disclosed
EP-1064273-A2 1,3,4-THIADIAZOLES USEFUL FOR THE TREATMENT OF CMV INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 2001-01-03 EP disclosed
US-6150385-A VIRICIDE WITH ACTIVITY AGAINST CYTOMEGALO VIRUS (CMV), HERPES VIRUS INCLUDING VARICELLA ZOSTER VIRUS, THE EPSTEIN-BARR VIRUS, THE HERPES SIMPLEX VIRUS, AND THE HUMAN HERPES VIRUS TYPE 8 (HHV-8) PHARMACIA & UPJOHN COMPANY (US) 2000-11-21 US disclosed
WO-1999047507-A2 1,3,4-THIADIAZOLES USEFUL FOR THE TREATMENT OF CMV INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1999-09-23 WO disclosed