SCHEMBL7546473

SCHEMBL7546473

CCC(=O)N(c1cnno1)C1CCN(Cc2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.51
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
OPRM1 P35372 5/20 0.50
SIGMAR1 Q99720 3/20 0.50
OPRD1 P41143 3/20 0.48
CHRM2 P08172 1/20 0.46
CHRM3 P20309 1/20 0.46
HRH3 Q9Y5N1 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MCHR1 Q99705 1/20 0.41
CXCR3 P49682 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7242607 0.79 OPRM1 (0.53) SMN1; SMN2KDM4EALDH1A1OPRM1SIGMAR1
SCHEMBL924276 0.74 OPRM1 (0.77) OPRM1SIGMAR1OPRD1CHRM2CHRM3
SCHEMBL3775423 0.72 OPRD1 (0.54) SMN1; SMN2KDM4EALDH1A1OPRM1SIGMAR1
SCHEMBL7487237 0.71 CHRM2 (0.65) SMN1; SMN2KDM4EALDH1A1SIGMAR1OPRD1
SCHEMBL20742038 0.68 OPRM1 (0.59) OPRM1SIGMAR1OPRD1CHRM3
SCHEMBL7487718 0.68 SIGMAR1 (0.74) SMN1; SMN2KDM4EALDH1A1SIGMAR1HRH3
SCHEMBL5744006 0.68 KDM4E (1.00) SMN1; SMN2KDM4EALDH1A1HRH3MEN1
SCHEMBL19501210 0.68 OPRM1 (0.62) OPRM1SIGMAR1OPRD1CHRM3
SCHEMBL6045571 0.68 OPRM1 (1.00) OPRM1SIGMAR1OPRD1CHRM2CHRM3
SCHEMBL4034421 0.68 KCNH2 (0.61) SMN1; SMN2KDM4EALDH1A1OPRM1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212299-A1 SUBSTITUTED PIPERIDINE COMPOUNDS USEFUL AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY AstraZeneca UK Limited (GB) 2002-06-12 EP disclosed
WO-2001014333-A1 SUBSTITUTED PIPERIDINE COMPOUNDS USEFUL AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY ASTRAZENECA UK LIMITED (GB) 2001-03-01 WO disclosed