SCHEMBL7546533

SCHEMBL7546533

CCCCNS(=O)(=O)Nc1ccc(-c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA14 Q9ULX7 1/20 0.48
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
NCOR2 Q9Y618 1/20 0.46
CA9 Q16790 2/20 0.44
PSEN1 P49768 1/20 0.44
PSEN2 P49810 1/20 0.44
APH1B Q8WW43 1/20 0.44
NCSTN Q92542 1/20 0.44
APH1A Q96BI3 1/20 0.44
PSENEN Q9NZ42 1/20 0.44
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
ALOX12 P18054 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19798391 0.90 CA1 (0.55) CA12CA1CA2CA7CA14
SCHEMBL29124111 0.84 PPARA (0.55) CA12CA1CA2CA7CA14
SCHEMBL7506954 0.79 KIF11 (0.40) CA12CA1CA2CA7CA14
SCHEMBL7506708 0.79 ACLY (0.44) CA12CA1CA2CA7CA14
SCHEMBL22558823 0.78 ALDH1A1 (0.63) CA12CA1CA2HDAC1HDAC2
SCHEMBL11526599 0.76 MAPT (0.54) CA12CA1CA2CA7CA14
SCHEMBL8972279 0.74 ALDH1A1 (0.56) HDAC3HDAC1HDAC2HDAC8NCOR2
SCHEMBL15444483 0.73 KEAP1 (0.42) CA12CA1CA2CA7CA14
SCHEMBL2930825 0.73 ALDH1A1 (0.64) CA12HDAC1HDAC2CA9GAA
SCHEMBL27945921 0.72 CA12 (0.69) CA12CA1CA2CA7CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216231-A2 INHIBITORS OF FACTOR Xa Millennium Pharmaceuticals, Inc. (US) 2002-06-26 EP disclosed
WO-2001019798-A2 INHIBITORS OF FACTOR Xa COR THERAPEUTICS INC. (US) 2001-03-22 WO disclosed