SCHEMBL7546596

SCHEMBL7546596

CC(C)(C)OC(=O)N1CCNCC1c1cccc(NC(=O)c2cccc(CCc3ccc(N)nc3)c2)c1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.40
PTK2 Q05397 2/20 0.36
RORC P51449 4/20 0.36
SCN9A Q15858 1/20 0.35
FLT4 P35916 1/20 0.34
ROCK2 O75116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7495243 0.91 RORC (0.37) HDAC1RORCSCN9A
SCHEMBL7546593 0.83 HDAC1 (0.36) HDAC1PTK2ROCK2
SCHEMBL6846514 0.80 TSHR (0.42) HDAC1
SCHEMBL6846512 0.71 PTPN11 (0.40) PTK2
Hydrochloric Acid SCHEMBL6844782 0.69 PTK2 (0.49) PTK2
SCHEMBL27909454 0.69 PARP1 (0.42) HDAC1
SCHEMBL30385469 0.69 PARP1 (0.42) HDAC1
SCHEMBL6844797 0.68 MET (0.39)
SCHEMBL30439890 0.67 TRPC6 (0.43)
SCHEMBL28505946 0.66 POLB (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252146-A1 AMIDE COMPOUNDS FOR INHIBITING PROTEIN KINASES AGOURON PHARMACEUTICALS, INC. (US) 2002-10-30 EP disclosed
WO-2001053274-A1 AMIDE COMPOUNDS FOR INHIBITING PROTEIN KINASES AGOURON PHARMACEUTICALS, INC. (US) 2001-07-26 WO disclosed