SCHEMBL7546982

SCHEMBL7546982

Nc1nccc(C(=O)c2cc(Cl)cc(Cl)c2Cl)c1C(=O)Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 6/20 0.36
SCN2A Q99250 4/20 0.36
SCN9A Q15858 3/20 0.36
SCN3A Q9NY46 3/20 0.36
SCN1A P35498 1/20 0.36
KCNH2 Q12809 1/20 0.36
SCN5A Q14524 1/20 0.36
RECQL P46063 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
CYP3A4 P08684 1/20 0.33
JAK2 O60674 2/20 0.32
TYK2 P29597 2/20 0.32
CDC7 O00311 1/20 0.32
PLK4 O00444 1/20 0.32
MAPK13 O15264 1/20 0.32
DAPK3 O43293 1/20 0.32
DYRK3 O43781 1/20 0.32
ROCK2 O75116 1/20 0.32
PRKD3 O94806 1/20 0.32
MAP4K4 O95819 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8804801 0.85 RECQL (0.46) RECQLL3MBTL1JAK2TYK2ALDH1A1
SCHEMBL8800986 0.79 RECQL (0.48) RECQLJAK2TYK2CDK2MAPK1
SCHEMBL7544426 0.78 HPGD (0.42) MAPK13MAPK12KDM4EMAPTALDH1A1
SCHEMBL7548664 0.77 KEAP1 (0.36) RECQLROCK2PRKD3MAP4K4LCK
SCHEMBL7549213 0.77 L3MBTL1 (0.41) RECQLL3MBTL1JAK2MAPK13KDR
SCHEMBL8805528 0.77 MAPK14 (0.40) RECQLL3MBTL1JAK2CDC7PLK4
SCHEMBL7549390 0.77 ALDH1A1 (0.50) CYP3A4JAK2TYK2CDK2ALDH1A1
SCHEMBL8799820 0.75 ALDH1A1 (0.40) KCNH2L3MBTL1MAPK13PRKCIMAPK12
SCHEMBL7546071 0.74 FLT1 (0.40) L3MBTL1JAK2MAPK13MAPK1KDR
SCHEMBL7547513 0.74 KMT2A (0.53) CYP3A4MAPK1KDRMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997049708-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1998-05-22 WO disclosed
WO-1996022295-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1996-11-14 WO disclosed