SCHEMBL7547161

SCHEMBL7547161

Cc1c(F)cccc1C(=O)c1ccnc(N)c1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 2/20 0.42
KDM4E B2RXH2 3/20 0.38
ASPH Q12797 1/20 0.38
KDM8 Q8N371 1/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
ALB P02768 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
TAS1R2 Q8TE23 1/20 0.36
KMT2A Q03164 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
DHODH Q02127 2/20 0.35
CDK2 P24941 1/20 0.35
MYC P01106 1/20 0.34
PRKCI P41743 1/20 0.33
PTPN1 P18031 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7553486 0.88 ALDH1A1 (0.37) NAPRTKDM4EASPHKDM8ESR1
SCHEMBL8813141 0.86 NAPRT (0.44) NAPRTKDM4EESR1ESR2KMT2A
SCHEMBL8802087 0.86 NAPRT (0.46) NAPRTKDM4EASPHKDM8KMT2A
SCHEMBL7553608 0.81 NAPRT (0.46) NAPRTKMT2ACYP3A4CYP2C9CDK2
SCHEMBL7548361 0.80 NAPRT (0.53) NAPRTKDM4EKMT2ACYP3A4CYP2C9
SCHEMBL8798744 0.79 NAPRT (0.44) NAPRTKDM4EASPHKDM8KMT2A
SCHEMBL7550390 0.76 KEAP1 (0.42) NAPRTKDM4EASPHKDM8ESR1
SCHEMBL7548942 0.76 KEAP1 (0.39) NAPRTKDM4EASPHKDM8KMT2A
SCHEMBL7548594 0.75 RECQL (0.48) NAPRTKMT2APRKCI
SCHEMBL8610741 0.75 CNR2 (0.50) NAPRTCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997049708-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1998-05-22 WO disclosed