SCHEMBL7548942

SCHEMBL7548942

Cc1cc(F)ccc1C(=O)c1ccnc(N)c1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.39
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
MAPK14 Q16539 4/20 0.38
MAPK13 O15264 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ASPH Q12797 1/20 0.38
KDM8 Q8N371 1/20 0.38
MAP4K4 O95819 1/20 0.38
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550390 0.90 KEAP1 (0.42) KEAP1TP53MAPK14KDM4EASPH
SCHEMBL7547613 0.85 PYGL (0.42) KEAP1MAPK14MAPK13MAPK12MAPK11
SCHEMBL7554905 0.84 L3MBTL1 (0.41) KDM4EGABRPGABRDGABRA1GABRB1
SCHEMBL7553546 0.82 KEAP1 (0.42) KEAP1TP53MAPK14KDM4EASPH
SCHEMBL7553608 0.81 NAPRT (0.46) MAPK14MAPK13MAPK12MAPK11NAPRT
SCHEMBL9059196 0.81 TP53 (0.38) KEAP1TP53MAPTMAPK14MAPK13
SCHEMBL7550244 0.78 MAPK14 (0.35) KEAP1TP53MAPK14MAPK13MAPK12
SCHEMBL7551790 0.78 SGMS2 (0.36) KEAP1TP53MAPTKDM4EASPH
SCHEMBL7547161 0.76 NAPRT (0.42) KDM4EASPHKDM8NAPRTDHODH
SCHEMBL7548264 0.76 KMO (0.43) MAPK14MAPK13MAPK12KDM4EASPH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997049708-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1998-05-22 WO disclosed