SCHEMBL8798744

SCHEMBL8798744

Cc1cccc(C)c1C(=O)c1ccnc(N)c1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.44
NOS3 P29474 3/20 0.41
NOS2 P35228 3/20 0.41
NOS1 P29475 1/20 0.41
KMT2A Q03164 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
MYC P01106 2/20 0.38
KDM4E B2RXH2 5/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KDM5A P29375 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
ASPH Q12797 1/20 0.36
KDM8 Q8N371 1/20 0.36
KDM4A O75164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8813141 0.87 NAPRT (0.44) NAPRTNOS3NOS2NOS1KMT2A
SCHEMBL7553608 0.87 NAPRT (0.46) NAPRTNOS3NOS2NOS1KMT2A
SCHEMBL1260539 0.80 NOS2 (0.52) NAPRTNOS3NOS2NOS1KMT2A
SCHEMBL7548361 0.79 NAPRT (0.53) NAPRTNOS3NOS2NOS1KMT2A
SCHEMBL7547161 0.79 NAPRT (0.42) NAPRTNOS3NOS2KMT2ACYP3A4
SCHEMBL7551656 0.78 TDP1 (0.39) NAPRTNOS3NOS2KMT2AL3MBTL1
SCHEMBL7547531 0.78 NAPRT (0.44) NAPRTNOS3NOS2NOS1KMT2A
SCHEMBL19857454 0.78 NAPRT (0.57) NAPRTKMT2AL3MBTL1TDP1CYP3A4
SCHEMBL8798672 0.77 RAB9A (0.42) NAPRTKMT2AL3MBTL1KDM4EKDM4C
SCHEMBL20520335 0.77 NAPRT (0.47) NAPRTNOS3NOS2KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811008-A1 BICYCLIC BENZAZEPINE DERIVATIVES AS VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1997-12-10 EP disclosed