SCHEMBL7547848

SCHEMBL7547848

N#CC1Cc2c(F)cccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.44
CHRNA4 P43681 2/20 0.44
CHRNA7 P36544 1/20 0.44
KDM4E B2RXH2 2/20 0.38
DRD2 P14416 3/20 0.37
DRD3 P35462 3/20 0.37
EEF2K O00418 1/20 0.35
KDM1A O60341 2/20 0.34
KDM1B Q8NB78 1/20 0.34
AADAT Q8N5Z0 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CUL4A Q13619 1/20 0.33
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
HTR5A P47898 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24482370 0.81 DRD2 (0.42) CHRNB2CHRNA4CHRNA7KDM4EDRD2
SCHEMBL3263345 0.78 GID4 (0.40) KDM4EKDM1AALDH1A1HTR2CHTR2B
SCHEMBL1721503 0.78 TRPM5 (0.42) KDM4EKDM1AAADATALDH1A1HPGD
SCHEMBL3032214 0.78 CUL4A (0.39) CHRNB2CHRNA4CUL4AHTR2CHTR2B
SCHEMBL7431326 0.68 GRIN2D (0.41) CHRNB2CHRNA4KDM1AHTR2CHTR2B
SCHEMBL1722308 0.68 GRIN2D (0.41) CHRNB2CHRNA4KDM1AHTR2CHTR2B
SCHEMBL30308765 0.68 GID4 (0.45) KDM4EDRD2KDM1AALDH1A1
SCHEMBL20478461 0.68 GID4 (0.45) KDM4EDRD2KDM1AALDH1A1
SCHEMBL12362682 0.68 CHRNB2 (0.44) CHRNB2CHRNA4CHRNA7DRD2DRD3
SCHEMBL20532511 0.67 KDM4E (0.47) CHRNB2CHRNA4KDM4EEEF2KALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0940386-B1 Benzocyclobutan compounds, their process for preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2002-05-22 EP disclosed
US-6107345-A ANTIDEPRESSANT; PSYCHOLOGICAL DISORDERS ADIR ET COMPAGNIE (FR) 2000-08-22 US disclosed
EP-0940386-A1 Benzocyclobutan compounds, their process for preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-09-08 EP disclosed