SCHEMBL7548604

SCHEMBL7548604

CNC(C)COCc1cccnc1C

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
FFAR1 O14842 1/20 0.38
MMP1 P03956 2/20 0.34
ADAM17 P78536 1/20 0.34
NMT1 P30419 2/20 0.33
P2RX7 Q99572 1/20 0.33
PTAFR P25105 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
DCPS Q96C86 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2608860 0.84 KDM4E (0.55) NPC1RAB9AKDM4EMAPTHTT
SCHEMBL14348152 0.74 FFAR1 (0.45) MAPTFFAR1NMT1P2RX7SMN1; SMN2
SCHEMBL7544675 0.73 CYP11B1 (0.36) CHRNB2CHRNA4
SCHEMBL27752600 0.72 FFAR1 (0.39) NPC1RAB9AKDM4EMAPTHTT
SCHEMBL14615243 0.71 KDM4E (0.49) NPC1RAB9AKDM4EMAPTHTT
SCHEMBL2084548 0.71 GABRA1 (0.47) NPC1KDM4EL3MBTL1FFAR1P2RX7
SCHEMBL7547886 0.71 CHRNB2 (0.46) CHRNB2CHRNA4
SCHEMBL7548586 0.71 MEN1 (0.38)
SCHEMBL7545392 0.71 CHRNB2 (0.46) CHRNB2CHRNA4
SCHEMBL12414712 0.70 FFAR1 (0.48) NPC1RAB9AKDM4EMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212301-A1 ARYLALKYLOXYALKYLAMINES AND ARYLALKYLTHIOALKYLAMINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS INHIBITORS OF NICOTINIC CHOLINERGIC RECEPTORS Targacept, Inc. (US) 2002-06-12 EP disclosed
WO-2001016107-A1 ARYLALKYLOXYALKYLAMINES AND ARYLALKYLTHIOALKYLAMINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS INHIBITORS OF NICOTINIC CHOLINERGIC RECEPTORS TARGACEPT, INC. (US) 2001-03-08 WO disclosed