SCHEMBL7549280

SCHEMBL7549280

O=c1[nH]nc(O)c2nc3ccc(F)cc3cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
TYMS P04818 3/20 0.39
DAO P14920 3/20 0.39
PARP1 P09874 3/20 0.39
KDM4E B2RXH2 1/20 0.36
BACE1 P56817 1/20 0.36
DDO Q99489 1/20 0.36
TSHR P16473 1/20 0.35
CASP3 P42574 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35
TUBB8 Q3ZCM7 1/20 0.35
TUBA3E Q6PEY2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550534 0.84 PDE3B (0.44) PDE3BPDE3ATYMSDAOPARP1
SCHEMBL7550176 0.84 CHEK1 (0.38) PDE3BPDE3ATYMSKDM4EBACE1
SCHEMBL7547477 0.82 KDM4E (0.44) PDE3BPDE3APARP1KDM4ECYP1A2
SCHEMBL7549332 0.76 CSNK2A1 (0.33) PDE3BPDE3ACYP1A2
SCHEMBL7545063 0.73 CSNK2A1 (0.35) CYP1A2
SCHEMBL7504185 0.70 DAO (0.36) PDE3BPDE3ATYMSDAOPARP1
SCHEMBL8872919 0.67 KDM4E (0.47) PDE3BPDE3ADAOKDM4EBACE1
SCHEMBL27171556 0.65 ERN1 (0.43) PDE3BPDE3ADAOKDM4EBACE1
SCHEMBL30984913 0.64 DAO (0.44) TYMSDAOPARP1KDM4EMAPT
SCHEMBL29655244 0.63 ALDH1A1 (0.56) TYMSDAOPARP1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0931081-B1 PYRIDAZINO 4,5-B]-QUINOLINE 5-OXIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS GLYCINE ANTAGONISTS MERZ & CO GMBH & CO (DE) 2002-09-25 EP claimed